2-piperidin-4-yl-benzimidazoles with broad spectrum antibacterial activities

Bioorg Med Chem Lett. 2003 Oct 6;13(19):3253-6. doi: 10.1016/s0960-894x(03)00661-9.

Abstract

A series of 2-piperidin-4-yl-benzimidazoles were synthesized and evaluated for antibacterial activities. Certain compounds inhibit bacterial growth with low micromolar minimal inhibitory concentration (MIC). These benzimidazoles are effective against both Gram-positive and Gram-negative bacteria of clinical importance, particularly enterococci, and represent a new class of potential antibacterial agents.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Anti-Bacterial Agents / chemistry*
  • Anti-Bacterial Agents / pharmacology
  • Benzimidazoles / chemistry*
  • Benzimidazoles / pharmacology
  • Enterococcus / drug effects
  • Enterococcus / growth & development
  • Microbial Sensitivity Tests / methods
  • Piperidines / chemistry*
  • Piperidines / pharmacology

Substances

  • Anti-Bacterial Agents
  • Benzimidazoles
  • Piperidines