Abstract
The c-Myc oncoprotein is a transcription factor that controls genes involved in cell growth, apoptosis and oncogenesis. We and others recently showed that the F-box protein Skp2 interacts with c-Myc and participates in its ubiquitylation and proteasomal degradation. Surprisingly, Skp2 was also found to act as a positive cofactor for c-Myc-regulated transcription. Further, Skp2, ubiquitylated proteins and subunits of the proteasome were demonstrated to be associated with a c-Myc target promoter in vivo. We show here that c-Myc interacts with Skp2 as part of the SCFSkp2 E3 ubiquitin ligase complex. Further, c-Myc interacts with the Sug1, an AAA ATPase subunit of the 19S regulatory particle of the proteasome. Inhibition of Sug1 expression by siRNA reduced transcription from a Myc target promoter to the same extent as c-Myc or Skp2 siRNA, implicating Sug1in this process. Taken together these findings suggest a role of the ubiquitin/proteasome system in c-Myc-regulated transcription. A hypothetical model discussing the link between ubiquitylation and transcription will be presented.
MeSH terms
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ATPases Associated with Diverse Cellular Activities
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Adaptor Proteins, Signal Transducing*
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Animals
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COS Cells
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Carrier Proteins / metabolism
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Cell Division / physiology
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Chlorocebus aethiops
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Cysteine Endopeptidases / metabolism*
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Intracellular Signaling Peptides and Proteins
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LIM Domain Proteins
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Multienzyme Complexes / metabolism*
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Promoter Regions, Genetic / physiology
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Proteasome Endopeptidase Complex
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Protein Interaction Mapping
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Proto-Oncogene Proteins c-myc / metabolism*
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S-Phase Kinase-Associated Proteins / metabolism*
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SKP Cullin F-Box Protein Ligases / metabolism
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Transcription Factors*
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Transcription, Genetic / genetics*
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Transcription, Genetic / physiology
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Ubiquitins / metabolism*
Substances
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Adaptor Proteins, Signal Transducing
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Carrier Proteins
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Intracellular Signaling Peptides and Proteins
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LIM Domain Proteins
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Multienzyme Complexes
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PSMC5 protein, human
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Proto-Oncogene Proteins c-myc
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S-Phase Kinase-Associated Proteins
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SUG1 protein, mammalian
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Transcription Factors
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Ubiquitins
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SKP Cullin F-Box Protein Ligases
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Cysteine Endopeptidases
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Proteasome Endopeptidase Complex
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ATPases Associated with Diverse Cellular Activities