2,5-Anhydro-D-mannitol increases hepatocyte calcium: implications for a hepatic hunger stimulus

Biochim Biophys Acta. 2003 Sep 23;1642(1-2):59-66. doi: 10.1016/s0167-4889(03)00099-5.

Abstract

The fructose analogue, 2,5-anhydro-D-mannitol (2,5-AM), triggers feeding in rats via a mechanism linked to its ability to trap phosphate and deplete hepatic ATP. This metabolic inhibitor is particularly useful in the study of the role of the liver in initiation of feeding as its effects are preferentially localized to the liver, and its metabolic consequences have been extensively characterized. To determine whether changes in intracellular calcium may participate in a mechanism conveying information about hepatic energy status to the nervous system, we studied the effects of 2,5-AM on intracellular calcium in isolated hepatocytes using the ratiometric indicator, fura-2. 2,5-AM elicited a marked elevation of intracellular calcium within 2-3 min of exposure that returned to baseline upon removal of the agent. Removal of external calcium failed to prevent this response, while emptying intracellular stores prevented it. These data are consistent with the hypothesis that hepatic energy status may be conveyed to the nervous system via a calcium-mediated secretion event.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Appetite Regulation / drug effects
  • Appetite Regulation / physiology
  • Calcium / deficiency
  • Calcium / metabolism*
  • Calcium Signaling / drug effects
  • Calcium Signaling / physiology
  • Energy Metabolism / drug effects
  • Energy Metabolism / physiology
  • Fluorescent Dyes
  • Fura-2
  • Hepatocytes / drug effects
  • Hepatocytes / metabolism*
  • Hunger / drug effects
  • Hunger / physiology*
  • Intracellular Fluid / drug effects
  • Intracellular Fluid / metabolism
  • Liver / cytology
  • Liver / drug effects
  • Liver / metabolism*
  • Male
  • Mannitol / analogs & derivatives*
  • Mannitol / pharmacology*
  • Rats
  • Signal Transduction / drug effects
  • Signal Transduction / physiology
  • Up-Regulation / drug effects
  • Up-Regulation / physiology

Substances

  • Fluorescent Dyes
  • Mannitol
  • 2,5-anhydromannitol
  • Calcium
  • Fura-2