Is the osteoclast calcium "receptor" a receptor-operated calcium channel?

Biochem Biophys Res Commun. 1992 Mar 16;183(2):619-25. doi: 10.1016/0006-291x(92)90527-r.

Abstract

Elevated extracellular calcium levels ([Ca2+]e) inhibit osteoclast function by elevating cytosolic free calcium levels ([Ca2+]i), presumably via the activation of a surface Ca2+ "receptor". It is unclear whether or not Ca(2+)-induced [Ca2+]i elevation involves the direct gating, by the putative "receptor", of a divalent cation channel. The results show that [Ca2+]i elevation in response to elevated [Ca2+]e comprises a distinct component of Ca2+ influx, the magnitude of which can be decreased and increased, respectively, by depolarising (100 mM-[K+]) and hyperpolarising (1 microM-[valinomycin]) the osteoclast membrane. In addition, activation of the putative Ca2+ "receptor" by elevated [Ca2+]e causes influx of the related divalent cation, magnesium (Mg2+). We suggest that Ca2+ influx induced by Ca2+ "receptor" activation is a major component of the observed [Ca2+]i response.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Animals, Newborn
  • Calcium / metabolism*
  • Calcium Channels / metabolism
  • Femur
  • Magnesium / metabolism
  • Membrane Potentials
  • Osteoclasts / drug effects
  • Osteoclasts / metabolism*
  • Potassium / pharmacology
  • Rats
  • Signal Transduction* / drug effects
  • Tibia
  • Valinomycin / pharmacology

Substances

  • Calcium Channels
  • Valinomycin
  • Magnesium
  • Potassium
  • Calcium