On the relationship between molecular mass and anticoagulant activity in a low molecular weight heparin (enoxaparin)

Thromb Haemost. 1992 May 4;67(5):556-62.

Abstract

A low molecular weight heparin (enoxaparin, mean molecular weight approximately 4,400) was separated by gel chromatography into eight different fractions with a narrow distribution around the following mean molecular weights: 1,800, 2,400, 2,900, 4,200, 6,200, 8,600, 9,800 and 11,000. We compared the influence of enoxaparin on the generation of thrombin in plasma to that of the eight fractions. We determined: a) the % of material with high affinity to antithrombin III (HAM) and the % of HAM above the critical chain length necessary to allow for thrombin inhibition (ACLM), b) the specific catalytic activity on the decay of endogenous thrombin, and c) the inhibition of over-all thrombin formation in the extrinsic and the intrinsic pathway. From b and c we calculated the inhibition of prothrombin conversion in these pathways. We found that a) there is a gradual decrease of the HAM fraction with decreasing molecular weight; b) the specific catalytic activity for the inactivation of thrombin does not vary significantly between the fractions when expressed in terms of ACLM; c) the potency to inhibit prothrombin conversion does not vary significantly between the fractions when expressed in terms of HAM.

Publication types

  • Comparative Study

MeSH terms

  • Antithrombin III / chemistry
  • Fluorescence
  • Heparin, Low-Molecular-Weight / chemistry
  • Heparin, Low-Molecular-Weight / pharmacology*
  • Humans
  • Molecular Weight
  • Thrombin / antagonists & inhibitors*
  • Thrombin / biosynthesis
  • Thromboplastin / antagonists & inhibitors*

Substances

  • Heparin, Low-Molecular-Weight
  • Antithrombin III
  • Thromboplastin
  • Thrombin