Human Y-79 retinoblastoma cells express functional corticotropin-releasing hormone receptors

Brain Res. 1992 Oct 16;593(2):304-6. doi: 10.1016/0006-8993(92)91324-8.

Abstract

In human Y-79 retinoblastoma cells corticotropin-releasing hormone (CRH) produces a marked and rapid increase of adenylate cyclase activity. The concentration of the peptide producing half-maximal stimulation is 60 nM. The effect of CRH is significantly antagonized by the specific CRH receptor antagonist alpha-helical CHR 9-41 and is mimicked by sauvagine and urotensin I, two peptides displaying sequence homology with CRH. These results demonstrate the presence of functional CRH receptors in human Y-79 retinoblastoma cells and suggest that this cell line may be a suitable model in which to study the action of CRH on human retinal cell function.

MeSH terms

  • Adenylyl Cyclases / metabolism*
  • Cell Line
  • Corticotropin-Releasing Hormone / antagonists & inhibitors
  • Corticotropin-Releasing Hormone / metabolism
  • Corticotropin-Releasing Hormone / pharmacology*
  • Eye Neoplasms
  • Humans
  • Kinetics
  • Peptide Fragments / pharmacology
  • Receptors, Corticotropin-Releasing Hormone
  • Receptors, Neurotransmitter / metabolism
  • Receptors, Neurotransmitter / physiology*
  • Retinoblastoma

Substances

  • Peptide Fragments
  • Receptors, Corticotropin-Releasing Hormone
  • Receptors, Neurotransmitter
  • Corticotropin-Releasing Hormone
  • corticotropin releasing hormone (9-41)
  • Adenylyl Cyclases