Atrial natriuretic peptide inhibits the spontaneous contractions of rabbit isolated ileum

J Pharm Pharmacol. 1992 Jul;44(7):615-7. doi: 10.1111/j.2042-7158.1992.tb05477.x.

Abstract

The present study investigates the effects of atriopeptin II on spontaneous phasic contractions of rabbit isolated ileum. Atriopeptin II caused a significant and concentration-dependent decrease in ileum motor activity. This effect was mimicked by 8-Br-cGMP and it was not affected by pretreatment with tetrodotoxin. Verapamil significantly decreased ileum contractions; however, in the presence of this calcium blocker, atriopeptin II further reduced ileal motility. These findings demonstrate that atriopeptin II depresses the motility of rabbit ileum through a cGMP-dependent mechanism and suggest that neither ileal neural networks nor extracellular calcium are involved in this effect.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Atrial Natriuretic Factor / pharmacology*
  • Dose-Response Relationship, Drug
  • Female
  • Ileum / drug effects*
  • In Vitro Techniques
  • Male
  • Muscle Contraction / drug effects*
  • Peptide Fragments
  • Rabbits

Substances

  • Peptide Fragments
  • Atrial Natriuretic Factor
  • atrial natriuretic factor prohormone (103-125)