In the GluR1 glutamate receptor subunit a glutamine to histidine point mutation suppresses inward rectification but not calcium permeability

Biochem Biophys Res Commun. 1992 Feb 14;182(3):1089-93. doi: 10.1016/0006-291x(92)91843-f.

Abstract

Recent papers have described glutamine to arginine point mutations of the cloned AMPA/Kainate receptor subunits that alter current-voltage relationship and suppress Ca2+ permeability, thus linking these two characteristics. We describe a glutamine to histidine mutation at the same position, which alters current-voltage relationship but retains Ca2+ permeability, thus dissociating the two properties.

MeSH terms

  • Animals
  • Barium / pharmacology
  • Base Sequence
  • Calcium / metabolism*
  • Calcium Channels / drug effects
  • Calcium Channels / physiology*
  • Cloning, Molecular
  • Evoked Potentials / drug effects
  • Glutamates / metabolism*
  • Glutamine*
  • Histidine*
  • Ibotenic Acid / analogs & derivatives
  • Ibotenic Acid / pharmacology
  • Kainic Acid / pharmacology
  • Macromolecular Substances
  • Molecular Sequence Data
  • Mutagenesis, Site-Directed*
  • Oligodeoxyribonucleotides
  • Oocytes / drug effects
  • Oocytes / physiology*
  • Plasmids
  • Quinoxalines / pharmacology
  • Receptors, Glutamate
  • Receptors, Neurotransmitter / genetics
  • Receptors, Neurotransmitter / metabolism
  • Receptors, Neurotransmitter / physiology*
  • Transcription, Genetic
  • Xenopus laevis
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid

Substances

  • Calcium Channels
  • Glutamates
  • Macromolecular Substances
  • Oligodeoxyribonucleotides
  • Quinoxalines
  • Receptors, Glutamate
  • Receptors, Neurotransmitter
  • Glutamine
  • Barium
  • Ibotenic Acid
  • Histidine
  • FG 9041
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid
  • Kainic Acid
  • Calcium