Effective alpha-particle-mediated radioimmunotherapy of murine leukemia

Cancer Res. 1992 Oct 15;52(20):5818-20.

Abstract

The specificity, toxicity, and efficacy of alpha-particle-mediated radioimmunotherapy of murine erythroleukemia was assessed by use of tumor-specific monoclonal antibody 103A labeled with 212Bi. Forty % of the injected dose/g tissue targeted to neoplastic spleens within 1 h after i.v. injection. When 212Bi-103A was injected on day 13 of disease, a dose-dependent response was achieved, as measured by a reduction in splenomegaly and absence of liver metastasis. Mice treated with 212Bi-103A on day 8 of disease showed no histological evidence of erythroleukemia on day 22 and survived significantly longer (median, 118 days) than mice treated with 212Bi-control IgG (78 days) or untreated mice (63 days), indicating successful specific radioimmunotherapy.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Alpha Particles / therapeutic use*
  • Animals
  • Antibodies, Monoclonal / therapeutic use*
  • Bismuth / pharmacokinetics
  • Bismuth / therapeutic use*
  • Cattle
  • Immunoglobulin G / therapeutic use
  • Mice
  • Radioimmunotherapy*
  • Radioisotopes / pharmacokinetics
  • Radioisotopes / therapeutic use*
  • Rauscher Virus

Substances

  • Antibodies, Monoclonal
  • Immunoglobulin G
  • Radioisotopes
  • Bismuth