Olvanil: more potent than capsaicin at stimulating the efferent function of sensory nerves

Eur J Pharmacol. 1992 Sep 4;219(3):481-4. doi: 10.1016/0014-2999(92)90494-o.

Abstract

The capsaicin analogue olvanil stimulated an increase in cutaneous blood flow when injected intradermally into the anaesthetised rabbit, as measured using a 133Xenon clearance method. Olvanil was found to be a 10-fold more potent vasodilator (on a molar basis) than capsaicin. The effect of both vasodilators was significantly inhibited by the calcitonin gene-related peptide (CGRP) receptor antagonist CGRP-(8-37). These findings suggest that olvanil stimulates the efferent function of cutaneous sensory nerves in a more potent manner than capsaicin. We therefore suggest that olvanil is a useful pharmacological tool for studying the activity of neuropeptides released from sensory nerves.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anesthesia
  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Blood Circulation / drug effects*
  • Calcitonin Gene-Related Peptide / metabolism
  • Capsaicin / analogs & derivatives*
  • Capsaicin / pharmacology*
  • Dose-Response Relationship, Drug
  • Efferent Pathways / drug effects
  • Injections, Intradermal
  • Neurons, Afferent / drug effects*
  • Rabbits
  • Xenon Radioisotopes

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Xenon Radioisotopes
  • olvanil
  • Calcitonin Gene-Related Peptide
  • Capsaicin