R2D2, a bridge between the initiation and effector steps of the Drosophila RNAi pathway

Science. 2003 Sep 26;301(5641):1921-5. doi: 10.1126/science.1088710.

Abstract

The RNA interference (RNAi) pathway is initiated by processing long double-stranded RNA into small interfering RNA (siRNA). The siRNA-generating enzyme was purified from Drosophila S2cells and consists of two stoichiometric subunits: Dicer-2(DCR-2) and a previously unknown protein that we named R2D2. R2D2 is homologous to the Caenorhabditis elegans RNAi protein RDE-4. Association with R2D2 does not affect the enzymatic activity of DCR-2. Rather, the DCR-2/R2D2 complex, but not DCR-2 alone, binds to siRNA and enhances sequence-specific messenger RNA degradation mediated by the RNA-initiated silencing complex (RISC). These results indicate that R2D2 bridges the initiation and effector steps of the Drosophila RNAi pathway by facilitating siRNA passage from Dicer to RISC.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Argonaute Proteins
  • Biotinylation
  • Caenorhabditis elegans / genetics
  • Caenorhabditis elegans / metabolism
  • Caenorhabditis elegans Proteins / chemistry
  • Cell Line
  • Chemical Precipitation
  • Drosophila Proteins / chemistry
  • Drosophila Proteins / genetics
  • Drosophila Proteins / isolation & purification*
  • Drosophila Proteins / metabolism*
  • Drosophila melanogaster / genetics*
  • Drosophila melanogaster / metabolism
  • Electrophoretic Mobility Shift Assay
  • Endoribonucleases / genetics
  • Endoribonucleases / isolation & purification
  • Endoribonucleases / metabolism*
  • Kinetics
  • Molecular Sequence Data
  • Mutation
  • Protein Structure, Tertiary
  • RNA Helicases / genetics
  • RNA Helicases / isolation & purification*
  • RNA Helicases / metabolism*
  • RNA Interference*
  • RNA, Double-Stranded / metabolism
  • RNA, Messenger / metabolism
  • RNA, Small Interfering / metabolism*
  • RNA-Binding Proteins / chemistry
  • RNA-Binding Proteins / genetics
  • RNA-Binding Proteins / isolation & purification
  • RNA-Binding Proteins / metabolism*
  • RNA-Induced Silencing Complex / isolation & purification
  • RNA-Induced Silencing Complex / metabolism
  • Recombinant Proteins / metabolism
  • Ribonuclease III

Substances

  • AGO2 protein, Drosophila
  • Argonaute Proteins
  • Caenorhabditis elegans Proteins
  • Drosophila Proteins
  • R2D2 protein, Drosophila
  • RDE-4 protein, C elegans
  • RNA, Double-Stranded
  • RNA, Messenger
  • RNA, Small Interfering
  • RNA-Binding Proteins
  • RNA-Induced Silencing Complex
  • Recombinant Proteins
  • DCR-2 protein, Drosophila
  • Endoribonucleases
  • Ribonuclease III
  • RNA Helicases