Conjugation of poor inhibitors with surface binding groups: a strategy to improve inhibition

Chem Commun (Camb). 2003 Sep 21:(18):2328-9. doi: 10.1039/b305179j.

Abstract

Conjugation of surface binding groups with inhibitors for carbonic anhydrase leads to the conversion of weak inhibitors to strong inhibitors.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Binding, Competitive
  • Carbonic Anhydrase Inhibitors / chemical synthesis
  • Carbonic Anhydrase Inhibitors / chemistry*
  • Carbonic Anhydrase Inhibitors / metabolism
  • Carbonic Anhydrases / metabolism
  • Catalysis
  • Histidine / chemistry*
  • Kinetics
  • Metals, Heavy / chemistry
  • Metals, Heavy / metabolism
  • Models, Chemical
  • Molecular Structure
  • Organometallic Compounds / chemistry
  • Organometallic Compounds / metabolism
  • Protein Binding
  • Sulfonamides / chemical synthesis
  • Sulfonamides / chemistry*
  • Sulfonamides / metabolism

Substances

  • Carbonic Anhydrase Inhibitors
  • Metals, Heavy
  • Organometallic Compounds
  • Sulfonamides
  • Histidine
  • Carbonic Anhydrases