Pharmacology of the 5-hydroxytryptamine-induced depolarization of the ferret vagus nerve in vitro

Eur J Pharmacol. 1992 Oct 6;221(1):157-60. doi: 10.1016/0014-2999(92)90786-4.

Abstract

Grease-gap recordings revealed that 5-hydroxytryptamine (5-HT) depolarized the ferret vagus nerve (pEC50 = 4.9). This response was mimicked by 2-methyl-5-HT and 1-phenylbiguanide, but not by 5-carboxamidotryptamine. Paroxetine (1 microM) or ketamine (10 microM) did not potentiate the response. Ketanserin (1 microM) did not reduce the depolarization, but four 5-HT3 receptor antagonists did. It is concluded that 5-HT depolarizes the ferret vagus nerve via 5-HT3 receptors, but these receptors may differ pharmacologically from those in other species.

MeSH terms

  • Animals
  • Dose-Response Relationship, Drug
  • Female
  • Ferrets
  • In Vitro Techniques
  • Membrane Potentials / drug effects
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Serotonin / drug effects
  • Serotonin / analogs & derivatives
  • Serotonin / pharmacology*
  • Tubocurarine / pharmacology
  • Vagus Nerve / drug effects*
  • Vagus Nerve / physiology

Substances

  • Receptors, Serotonin
  • Serotonin
  • 2-methyl-5-HT
  • Tubocurarine