Solution structure and stability of a disulfide cross-linked nucleopeptide duplex

Chem Commun (Camb). 2003 Oct 21:(20):2558-9. doi: 10.1039/b307300a.

Abstract

NMR methods are used to study the structure and stability of the duplex formed by the nucleopeptide [Ac-Cys-Gly-Ala-Hse(p3'dGCATGC)-Ala-OH]2[S-S], in which the oligonucleotide is self-complementary and the cysteine residues of the two peptide chains form a disulfide bridge; thermal transitions and NMR-derived structural calculations are consistent with a 3-D structure in which the oligonucleotide forms a standard B-DNA helix without significant distortions; the peptide chains are relatively disordered in solution and lie in the minor groove of the DNA helix; this nucleopeptide duplex exhibits a high melting temperature, indicating that peptide-oligonucleotide conjugates containing cysteines are suitable molecules to establish cross-links between DNA strands and stabilize the duplex.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Base Sequence
  • Cysteine / chemistry
  • Disulfides / chemistry*
  • Models, Molecular
  • Molecular Structure
  • Nuclear Magnetic Resonance, Biomolecular
  • Nucleic Acid Conformation
  • Nucleic Acid Denaturation
  • Nucleoproteins / chemistry*
  • Oligonucleotides / chemistry
  • Protein Conformation
  • Solutions / chemistry
  • Temperature

Substances

  • Disulfides
  • Nucleoproteins
  • Oligonucleotides
  • Solutions
  • Cysteine