Crystal structure of a beta-catenin/axin complex suggests a mechanism for the beta-catenin destruction complex

Genes Dev. 2003 Nov 15;17(22):2753-64. doi: 10.1101/gad.1142603. Epub 2003 Nov 4.

Abstract

The "beta-catenin destruction complex" is central to canonical Wnt/beta-catenin signaling. The scaffolding protein Axin and the tumor suppressor adenomatous polyposis coli protein (APC) are critical components of this complex, required for rapid beta-catenin turnover. We determined the crystal structure of a complex between beta-catenin and the beta-catenin-binding domain of Axin (Axin-CBD). The Axin-CBD forms a helix that occupies the groove formed by the third and fourth armadillo repeats of beta-catenin and thus precludes the simultaneous binding of other beta-catenin partners in this region. Our biochemical studies demonstrate that, when phosphorylated, the 20-amino acid repeat region of APC competes with Axin for binding to beta-catenin. We propose that a key function of APC in the beta-catenin destruction complex is to remove phosphorylated beta-catenin product from the active site.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenomatous Polyposis Coli Protein / chemistry
  • Adenomatous Polyposis Coli Protein / metabolism
  • Amino Acid Sequence
  • Animals
  • Axin Protein
  • Binding Sites
  • Crystallography, X-Ray
  • Cytoskeletal Proteins / chemistry*
  • Cytoskeletal Proteins / metabolism
  • Humans
  • Models, Molecular
  • Molecular Sequence Data
  • Phosphorylation
  • Protein Binding
  • Protein Conformation
  • Proteins / chemistry*
  • Proteins / metabolism
  • Repressor Proteins*
  • Sequence Homology, Amino Acid
  • Signal Transduction
  • Trans-Activators / chemistry*
  • Trans-Activators / metabolism
  • Xenopus Proteins
  • Xenopus laevis / metabolism
  • beta Catenin

Substances

  • Adenomatous Polyposis Coli Protein
  • Axin Protein
  • CTNNB1 protein, Xenopus
  • CTNNB1 protein, human
  • Cytoskeletal Proteins
  • Proteins
  • Repressor Proteins
  • Trans-Activators
  • Xenopus Proteins
  • axin1 protein, Xenopus
  • beta Catenin