IL-7-dependent human leukemia T-cell line as a valuable tool for drug discovery in T-ALL

Blood. 2004 Mar 1;103(5):1891-900. doi: 10.1182/blood-2002-12-3861. Epub 2003 Nov 13.

Abstract

The specific targeting of critical signaling molecules may provide efficient therapies for T-cell acute lymphoblastic leukemia (T-ALL). However, target identification and drug development are limited by insufficient numbers of primary T-ALL cells and by their high rate of spontaneous apoptosis. We established a human interleukin-7 (IL-7)-dependent T-ALL cell line, TAIL7, that maintains several biologic and signaling properties of its parental leukemia cells. TAIL7 cells are pre-T-ALL cells that proliferate in response to IL-7 and IL-4. IL-7 stimulation of TAIL7 cells prevents spontaneous in vitro apoptosis and induces cell activation and cell cycle progression. The signaling events triggered by IL-7 include down-regulation of p27(kip1) and hyperphosphorylation of retinoblastoma protein (Rb). Stimulation of TAIL7 cells by IL-7 leads to phosphorylation of Janus kinase 3 (JAK3), signal transducer and activator of transcription 5 (STAT5), Akt/PKB (protein kinase B), and extracellular-regulated kinase 1 and 2 (Erk1/2). Importantly, specific blockade of JAK3 by its inhibitor WHI-P131 abrogates the IL-7-mediated proliferation and survival of TAIL7 cells, suggesting that activation of JAK3 is critical for IL-7 responsiveness by these cells. Because TAIL7 cells seem to be a biologic surrogate for primary leukemia T cells, this cell line constitutes a valuable tool for the study of the signaling pathways implicated in T-ALL. Exploitation of this cell line should allow the identification of molecular targets and promote the rational design and validation of antileukemia signaling inhibitors.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Cell Cycle
  • Cell Cycle Proteins / metabolism
  • Cell Division
  • Cell Line, Tumor*
  • Cell Survival
  • Cyclin-Dependent Kinase Inhibitor p27
  • DNA / metabolism
  • Disease Progression
  • Down-Regulation
  • Enzyme Activation
  • Humans
  • Immunoblotting
  • Immunophenotyping
  • Interleukin-4 / metabolism
  • Interleukin-7 / genetics*
  • Interleukin-7 / metabolism
  • Janus Kinase 3
  • Karyotyping
  • Leukemia-Lymphoma, Adult T-Cell / metabolism*
  • Mice
  • Mice, Inbred NOD
  • Mice, SCID
  • Mitogen-Activated Protein Kinase 1 / metabolism
  • Mitogen-Activated Protein Kinase 3
  • Mitogen-Activated Protein Kinases / metabolism
  • Phenotype
  • Phosphorylation
  • Precipitin Tests
  • Protein-Tyrosine Kinases / metabolism
  • Retinoblastoma Protein / metabolism
  • Reverse Transcriptase Polymerase Chain Reaction
  • Signal Transduction
  • T-Lymphocytes / metabolism*
  • Tumor Suppressor Proteins / metabolism

Substances

  • Cdkn1b protein, mouse
  • Cell Cycle Proteins
  • Interleukin-7
  • Retinoblastoma Protein
  • Tumor Suppressor Proteins
  • Cyclin-Dependent Kinase Inhibitor p27
  • Interleukin-4
  • DNA
  • Protein-Tyrosine Kinases
  • JAK3 protein, human
  • Jak3 protein, mouse
  • Janus Kinase 3
  • Mitogen-Activated Protein Kinase 1
  • Mitogen-Activated Protein Kinase 3
  • Mitogen-Activated Protein Kinases