Snail mediates E-cadherin repression by the recruitment of the Sin3A/histone deacetylase 1 (HDAC1)/HDAC2 complex

Mol Cell Biol. 2004 Jan;24(1):306-19. doi: 10.1128/MCB.24.1.306-319.2004.

Abstract

The transcription factor Snail has been described as a direct repressor of E-cadherin expression during development and carcinogenesis; however, the specific mechanisms involved in this process remain largely unknown. Here we show that mammalian Snail requires histone deacetylase (HDAC) activity to repress E-cadherin promoter and that treatment with trichostatin A (TSA) is sufficient to block the repressor effect of Snail. Moreover, overexpression of Snail is correlated with deacetylation of histones H3 and H4 at the E-cadherin promoter, and TSA treatment in Snail-expressing cells reverses the acetylation status of histones. Additionally, we demonstrate that Snail interacts in vivo with the E-cadherin promoter and recruits HDAC activity. Most importantly, we demonstrate an interaction between Snail, histone deacetylase 1 (HDAC1) and HDAC2, and the corepressor mSin3A. This interaction is dependent on the SNAG domain of Snail, indicating that the Snail transcription factor mediates the repression by recruitment of chromatin-modifying activities, forming a multimolecular complex to repress E-cadherin expression. Our results establish a direct causal relationship between Snail-dependent repression of E-cadherin and the modification of chromatin at its promoter.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cadherins / metabolism*
  • DNA-Binding Proteins / metabolism*
  • Gene Expression Regulation
  • Histone Deacetylase 2
  • Histone Deacetylases / metabolism*
  • Humans
  • Mice
  • Promoter Regions, Genetic
  • Repressor Proteins / metabolism*
  • Sin3 Histone Deacetylase and Corepressor Complex
  • Snail Family Transcription Factors
  • Transcription Factors / metabolism*

Substances

  • Cadherins
  • DNA-Binding Proteins
  • Repressor Proteins
  • SIN3A transcription factor
  • Snail Family Transcription Factors
  • Transcription Factors
  • Hdac2 protein, mouse
  • Histone Deacetylase 2
  • Histone Deacetylases
  • Sin3 Histone Deacetylase and Corepressor Complex