A continuous assay of myristoyl-CoA:protein N-myristoyltransferase for proteomic analysis

Anal Biochem. 2003 Nov 1;322(1):116-23. doi: 10.1016/j.ab.2003.07.007.

Abstract

Protein N-myristoylation is an important lipid modification that affects the activity and membrane-binding properties of crucial proteins belonging to signal transduction cascades. The aim of this work was to develop a rapid and easy diagnostic method to check for (i) effective N-myristoylation of any given protein and (ii) easy proteome annotation. The N-myristoylation reaction was coupled to that of pyruvate dehydrogenase, and NADH was continuously detected spectrophotometrically. This method was optimized for and applied to full-length Saccharomyces cerevisiae and Arabidopsis thaliana N-myristoyltransferases and two A. thaliana enzyme derivatives. The data were validated by comparison with a previously described discontinuous assay, modification of the chemical nature of the substrates, and use of specific inhibitors. The kinetics of N-myristoylation were determined in vitro with various compounds including a full-length polypeptide substrate, a small G protein of the RAB family already known to be N-myristoylated in vivo. This automated assay can be used for proteomic studies to determine the N-myristoylation state of any protein.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acyl Coenzyme A / metabolism*
  • Acyltransferases / metabolism*
  • Arabidopsis / enzymology
  • Chromogenic Compounds / chemical synthesis
  • Cloning, Molecular
  • Ketone Oxidoreductases / metabolism
  • Myristic Acid / metabolism
  • Myristic Acids / metabolism
  • NADP / metabolism
  • Protein Conformation
  • Protein Processing, Post-Translational*
  • Proteomics
  • Recombinant Proteins / isolation & purification
  • Recombinant Proteins / metabolism
  • Saccharomyces cerevisiae / enzymology
  • Signal Transduction
  • Spectrum Analysis

Substances

  • Acyl Coenzyme A
  • Chromogenic Compounds
  • Myristic Acids
  • Recombinant Proteins
  • Myristic Acid
  • alpha-hydroxymyristic acid
  • S-tetradecanoyl-coenzyme A
  • NADP
  • Ketone Oxidoreductases
  • pyruvate dehydrogenase (NADP+)
  • Acyltransferases
  • glycylpeptide N-tetradecanoyltransferase