Temperature-dependent substrate inhibition of the cysteine proteinase (GP57/51) from Trypanosoma cruzi

Mol Biochem Parasitol. 1992 Dec;56(2):335-8. doi: 10.1016/0166-6851(92)90183-k.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antigens, Protozoan / metabolism*
  • Coumarins / pharmacology
  • Cysteine Endopeptidases / drug effects
  • Cysteine Endopeptidases / metabolism*
  • Cysteine Proteinase Inhibitors / pharmacology*
  • Dipeptides / pharmacology
  • Dose-Response Relationship, Drug
  • Glycoproteins / antagonists & inhibitors
  • Glycoproteins / metabolism*
  • Hot Temperature
  • Hydrogen-Ion Concentration
  • Hydrolysis
  • Trypanosoma cruzi / enzymology*

Substances

  • Antigens, Protozoan
  • Coumarins
  • Cysteine Proteinase Inhibitors
  • Dipeptides
  • Glycoproteins
  • benzyloxycarbonyl-phenylalanylarginine-4-methylcoumaryl-7-amide
  • benzyloxycarbonylarginyl-arginine 4-methylcoumarin-7-ylamide
  • Cysteine Endopeptidases
  • GP57-51 antigen, Trypanosoma cruzi