Quantification of percutaneous absorption of metronidazole and levamisole in the fire-bellied toad (Bombina orientalis)

J Vet Pharmacol Ther. 1992 Dec;15(4):433-6. doi: 10.1111/j.1365-2885.1992.tb01035.x.

Abstract

Spot-on application has proved to be an effective way to reach therapeutic doses of metronidazole and levamisole in fire-bellied toads. The percutaneous absorption of metronidazole and levamisole was quantified, using an aqueous solution of 1.008 mg/ml of metronidazole and an aqueous solution of 3.767 mg/ml of levamisole. High Performance Liquid Chromatography (HPLC) analysis of the percutaneous absorption revealed that of the amount applied, 75% of metronidazole and 90% of levamisole was absorbed. This resulted during 3 days of application in dosages of 23 mg/kg BW of metronidazole and 94 mg/kg BW of levamisole. Of the absorbed substances, 48% of metronidazole and 9% of levamisole were excreted in urine and faeces as unmetabolised substances.

MeSH terms

  • Administration, Cutaneous
  • Animals
  • Anura / metabolism*
  • Chromatography, High Pressure Liquid
  • Levamisole / pharmacokinetics*
  • Metronidazole / pharmacokinetics*
  • Skin Absorption*

Substances

  • Metronidazole
  • Levamisole