Photodynamic therapy of intestinal tumors with mono-L-aspartyl chlorin e6 (NPe6): a basic study

Anticancer Res. 2003 Nov-Dec;23(6C):4897-900.

Abstract

Background: To clarify the usefulness of the second-generation photosensitizer, mono-L-aspartyl chlorin e6 (NPe6), we examined the possibility of photodynamic diagnosis and photodynamic therapy for intestinal tumors in a mouse model.

Materials and methods: NPe6 was intravenously administered to the tumor-bearing mice through the tail vein. The intestinal tumor sites were irradiated with a 664-nm diode laser at constant intervals after the administration of photosensitizers. The tumors were excised and fluorescence was observed in frozen sections by microscope.

Results: We observed the fluorescent image and calculated that the mean fluorescence intensity was significantly higher in the tumors than the normal mucosa during 6 hours (p < 0.05). The fluorescence of NPe6 was chiefly accumulated in the intestinal tumors as red fluorescence on the fluorescent microphotographic image.

Conclusion: We conclude that NPe6 may be a valuable photosensitizer for the photodynamic diagnosis and photodynamic therapy of intestinal tumors.

MeSH terms

  • Animals
  • Disease Models, Animal
  • Intestinal Neoplasms / drug therapy*
  • Intestinal Neoplasms / pathology
  • Lasers
  • Mice
  • Mice, Inbred C57BL
  • Mice, Inbred Strains
  • Microscopy, Fluorescence
  • Photochemotherapy / methods*
  • Photosensitizing Agents / therapeutic use*
  • Porphyrins / therapeutic use*

Substances

  • Photosensitizing Agents
  • Porphyrins
  • Talaporfin