mTOR-dependent activation of the transcription factor TIF-IA links rRNA synthesis to nutrient availability

Genes Dev. 2004 Feb 15;18(4):423-34. doi: 10.1101/gad.285504.

Abstract

In cycling cells, transcription of ribosomal RNA genes by RNA polymerase I (Pol I) is tightly coordinated with cell growth. Here, we show that the mammalian target of rapamycin (mTOR) regulates Pol I transcription by modulating the activity of TIF-IA, a regulatory factor that senses nutrient and growth-factor availability. Inhibition of mTOR signaling by rapamycin inactivates TIF-IA and impairs transcription-initiation complex formation. Moreover, rapamycin treatment leads to translocation of TIF-IA into the cytoplasm. Rapamycin-mediated inactivation of TIF-IA is caused by hypophosphorylation of Se 44 (S44) and hyperphosphorylation of Se 199 (S199). Phosphorylation at these sites affects TIF-IA activity in opposite ways, for example, phosphorylation of S44 activates and S199 inactivates TIF-IA. The results identify a new target formTOR-signaling pathways and elucidate the molecular mechanism underlying mTOR-dependent regulation of RNA synthesis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3T3 Cells
  • Amino Acid Substitution
  • Animals
  • Cell Division
  • Cell Line
  • Cell Nucleus / metabolism
  • Humans
  • Mice
  • Mutagenesis, Site-Directed
  • Nucleic Acid Hybridization
  • Phosphates / metabolism
  • Phosphorylation
  • Pol1 Transcription Initiation Complex Proteins
  • Protein Kinases / metabolism*
  • Protein Transport
  • RNA Polymerase I / metabolism
  • RNA, Ribosomal / genetics*
  • Signal Transduction / drug effects
  • Sirolimus / pharmacology
  • TOR Serine-Threonine Kinases
  • Transcription Factors / chemistry
  • Transcription Factors / genetics
  • Transcription Factors / metabolism*
  • Transcription, Genetic / drug effects
  • Transcription, Genetic / genetics

Substances

  • Phosphates
  • Pol1 Transcription Initiation Complex Proteins
  • RNA, Ribosomal
  • RRN3 protein, human
  • Transcription Factors
  • Protein Kinases
  • MTOR protein, human
  • mTOR protein, mouse
  • TOR Serine-Threonine Kinases
  • RNA Polymerase I
  • Sirolimus