Biotransformation of triptolide and triptonide by cell suspension cultures of Catharanthus roseus

J Asian Nat Prod Res. 2004 Jun;6(2):93-7. doi: 10.1080/1028602031000135567.

Abstract

Catharanthus roseus cell suspension cultures were used to bioconvert both triptolide (1) and triptonide (2). The same reaction path was followed in both biotransformations. Two biotransformed products were obtained and their structures identified as triptriolide (3) and 12beta,13alpha-dihydroxytriptonide (4), respectively, from 1 and 2. Product 4 is a new compound.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biotransformation
  • Catharanthus / cytology
  • Catharanthus / metabolism*
  • Cells, Cultured
  • Diterpenes / pharmacokinetics*
  • Epoxy Compounds
  • Phenanthrenes / pharmacokinetics*
  • Triterpenes / pharmacokinetics*

Substances

  • Diterpenes
  • Epoxy Compounds
  • Phenanthrenes
  • Triterpenes
  • triptolide
  • triptonide