Ex vivo and in vivo biological effects of a truncated form of the receptor tyrosine kinase stk when activated by interaction with the friend spleen focus-forming virus envelope glycoprotein or by point mutation

J Virol. 2004 May;78(9):4573-81. doi: 10.1128/jvi.78.9.4573-4581.2004.

Abstract

The erythroleukemia-inducing Friend spleen focus-forming virus (SFFV) encodes a unique envelope protein, gp55, which interacts with the erythropoietin (Epo) receptor complex, causing proliferation and differentiation of erythroid cells in the absence of Epo. Susceptibility to SFFV-induced erythroleukemia is conferred by the Fv-2 gene, which encodes a short form of the receptor tyrosine kinase Stk/Ron (sf-Stk) only in susceptible strains of mice. We recently demonstrated that sf-Stk becomes activated by forming a strong interaction with SFFV gp55. To examine the biological consequences of activated sf-Stk on erythroid cell growth, we prepared retroviral vectors which express sf-Stk, either in conjunction with gp55 or alone in a constitutively activated mutant form, and tested them for their ability to induce Epo-independent erythroid colonies ex vivo and disease in mice. Our data indicate that both gp55-activated sf-Stk and the constitutively activated mutant of sf-Stk induce erythroid cells from Fv-2-susceptible and Fv-2-resistant (sf-Stk null) mice to form Epo-independent colonies. Mutational analysis of sf-Stk indicated that a functional kinase domain and 8 of its 12 tyrosine residues are required for the induction of Epo-independent colonies. Further studies demonstrated that coexpression of SFFV gp55 with sf-Stk significantly extends the half-life of the kinase. When injected into Fv-2-resistant mice, neither the gp55-activated sf-Stk nor the constitutively activated mutant caused erythroleukemia. Surprisingly, both Fv-2-susceptible and -resistant mice injected with the gp55-sf-Stk vector developed clinical signs not previously associated with SFFV-induced disease. We conclude that sf-Stk, activated by either point mutation or interaction with SFFV gp55, is sufficient to induce Epo-independent erythroid colonies from both Fv-2-susceptible and -resistant mice but is unable to cause erythroleukemia in Fv-2-resistant mice.

MeSH terms

  • Animals
  • Cell Line
  • Erythroid Cells / cytology
  • Erythroid Cells / metabolism*
  • Erythropoietin / metabolism
  • Genetic Vectors
  • Leukemia, Erythroblastic, Acute / physiopathology
  • Leukemia, Erythroblastic, Acute / virology
  • Mice
  • Mice, Inbred C57BL
  • Point Mutation*
  • Receptor Protein-Tyrosine Kinases / genetics
  • Receptor Protein-Tyrosine Kinases / metabolism*
  • Retroviridae Infections / physiopathology
  • Retroviridae Infections / virology
  • Spleen Focus-Forming Viruses / metabolism
  • Spleen Focus-Forming Viruses / pathogenicity*
  • Tumor Virus Infections / physiopathology
  • Tumor Virus Infections / virology
  • Viral Envelope Proteins / metabolism*

Substances

  • Viral Envelope Proteins
  • glycoprotein gp55, Friend spleen focus-forming virus
  • Erythropoietin
  • RON protein
  • Receptor Protein-Tyrosine Kinases