Solid-phase syntheses of furopyridine and furoquinoline systems

Org Lett. 2004 Apr 29;6(9):1405-8. doi: 10.1021/ol049762f.

Abstract

[reaction: see text] Syntheses of 2-substituted furo[3,2-b]pyridines and furo[3,2-h]quinolines have been achieved for the first time in the solid-phase mode. The central enabling steps involved concomitant deprotection/cyclization promoted by the mild base K(2)CO(3). Reactions were monitored "in situ" in real time by a variety of spectroscopic techniques, which allowed full and accurate control of progress in these syntheses.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Molecular Conformation
  • Pyridines / chemical synthesis*
  • Pyridines / chemistry
  • Quinolines / chemical synthesis*
  • Quinolines / chemistry

Substances

  • Pyridines
  • Quinolines