Photochemical preparation of 1,3,5,7-tetracyanoadamantane and its conversion to 1,3,5,7-tetrakis(aminomethyl)adamantane

Org Lett. 2004 May 27;6(11):1705-7. doi: 10.1021/ol036526g.

Abstract

New adamantane derivatives 1 and 2 that bear functionalized one-carbon extensions at all four bridgehead positions have been prepared. Radical nucleophilic substitution (S(RN)1) reaction of 1,3,5,7-tetrabromoadamantane with cyanide produces 1,3,5,7-tetracyanoadamantane (1), which was reduced with borane reagents to 1,3,5,7-tetrakis(aminomethyl)adamantane (2). Improvements in the preparation of 1,3,5,7-tetrahaloadamantanes (halogen = Br, Cl, I) are also reported. [structure--see text]

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adamantane / analogs & derivatives
  • Adamantane / chemistry*
  • Magnetic Resonance Spectroscopy
  • Molecular Structure
  • Photochemistry

Substances

  • 1,3,5,7-tetracyanoadamantane
  • 1,3,5,7-tetrakis(aminomethyl)adamantane
  • Adamantane