Field potential analysis in the freely moving rat during the action of cyclandelate or flunarizine

Pharmacol Res. 1992 Apr;25(3):287-97. doi: 10.1016/s1043-6618(05)80078-7.

Abstract

Cyclandelate and flunarizine, two vasoactive Ca2+ channel or Ca2+ overload blockers have been compared with respect to their in vivo action on field potentials recorded from the depths of the brain in freely moving rats. Whereas cyclandelate showed a dose dependent rapid onset of action in the range of 15 to 120 mg/kg i.p., flunarizine only induced weak effects very slowly, not reaching statistical relevance before the fourth hour after the injection (0.1 to 1.6 mg/kg). Even then no clear dose dependence could be recognized for flunarizine. With respect to the frequency content of the recorded signals a rather close similarity between both drugs could be seen. Comparison of the drug effects to our reference data base of more than 80 compounds revealed a close relationship to memantine, an antiparkinson drug, suspected to act on the NMDA (N-methyl-d-aspartate) receptor-ionophor complex controlling Ca2+ fluxes. There is some indication that cyclandelate might also act in a similar way at the molecular level.

MeSH terms

  • Administration, Oral
  • Animals
  • Brain / drug effects*
  • Brain / physiology
  • Calcium Channel Blockers / pharmacology*
  • Cyclandelate / pharmacology*
  • Dose-Response Relationship, Drug
  • Flunarizine / pharmacology*
  • Fourier Analysis
  • Injections, Intraperitoneal
  • Male
  • Membrane Potentials / drug effects
  • Multivariate Analysis
  • Rats
  • Rats, Inbred F344

Substances

  • Calcium Channel Blockers
  • Cyclandelate
  • Flunarizine