Influence of a lipase inhibitor on gastric sensitivity and accommodation to an orally ingested meal

Aliment Pharmacol Ther. 2004 Jun 15;19(12):1261-8. doi: 10.1111/j.1365-2036.2004.02003.x.

Abstract

Background: Intraduodenal administration of lipids, through lipid digestion and release of cholecystokinin (CCK), induces viscero-visceral reflexes that affect gastric tone and sensitivity. It is unclear whether the same mechanisms control gastric function after an orally ingested meal.

Aim: To evaluate the effect of orlistat, a selective lipase inhibitor, on gastric response to an orally administered meal.

Methods: Eighteen healthy volunteers participated in this study. They were treated for 5 days with orlistat (120 mg) or placebo t.d.s. in a double-blind randomized crossover design. During treatment, all subjects underwent a gastric barostat study, measurement of plasma CCK levels and a satiety drinking test.

Results: Although CCK plasma levels were significantly decreased, pre-treatment with orlistat failed to affect gastric compliance (72 +/- 6 mL/mm Hg and 64 +/- 6 mL/mm Hg, NS), gastric sensitivity (discomfort threshold 12.2 +/- 0.6 mm Hg vs. 10.9 +/- 0.6 mm Hg above minimal distending pressure, NS) or gastric accommodation (172 +/- 41 mL vs. 206 +/- 49 mL, NS) to an orally ingested meal. Furthermore, orlistat pre-treatment had no significant effect on the amount of calories ingested during a satiety drinking test (1329 +/- 88 kcal vs. 1217 +/- 115 kcal, NS).

Conclusion: Administration of a lipase inhibitor does not affect gastric compliance, sensitivity to distension and accommodation to an orally ingested meal, and does not influence meal-induced satiety.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial

MeSH terms

  • Adaptation, Physiological / physiology
  • Adolescent
  • Adult
  • Anti-Obesity Agents / pharmacology
  • Cholecystokinin / blood
  • Cross-Over Studies
  • Double-Blind Method
  • Eating / physiology*
  • Enzyme Inhibitors / pharmacology*
  • Fasting / physiology
  • Female
  • Gastric Emptying / drug effects
  • Humans
  • Lactones / pharmacology*
  • Lipase / antagonists & inhibitors*
  • Male
  • Orlistat
  • Postprandial Period / physiology
  • Pressure
  • Satiation / drug effects
  • Stomach / drug effects*
  • Stomach / physiology

Substances

  • Anti-Obesity Agents
  • Enzyme Inhibitors
  • Lactones
  • Cholecystokinin
  • Orlistat
  • Lipase