Synthesis and biological evaluation of novel apio nucleosides with thiazole-4-carboxamide and 1,2,4-triazole-3-carboxamide

Nucleosides Nucleotides Nucleic Acids. 2004;23(4):715-24. doi: 10.1081/NCN-120037666.

Abstract

In view of biological activities of azole nucleosides and apio-dideoxynucleoside, novel apio nucleoside analogues (1 and 2) with thiazole and triazole base moiety were synthesized using 2,3-O-isopropylidene-apio-beta-D-furanose (3), which was prepared from D-mannose.

MeSH terms

  • Mannose / analogs & derivatives*
  • Mannose / chemistry
  • Nucleosides / chemical synthesis*
  • Nucleosides / chemistry
  • Structure-Activity Relationship
  • Thiazoles / chemical synthesis*
  • Thiazoles / chemistry
  • Triazoles / chemical synthesis*
  • Triazoles / chemistry

Substances

  • Nucleosides
  • Thiazoles
  • Triazoles
  • Mannose