Expression of the sodium channel beta3 subunit in injured human sensory neurons

Neuroreport. 2004 Jul 19;15(10):1629-32. doi: 10.1097/01.wnr.0000134927.02776.ae.

Abstract

Voltage-gated sodium channel alpha-subunits play a key role in pain pathophysiology, and are modulated by beta-subunits. We previously reported that beta1- and beta2-subunits were decreased in human sensory neurons after spinal root avulsion injury. We have now detected, by immunohistochemistry, beta3-subunits in 82% of small/medium and 67% of large diameter sensory neurons in intact human dorsal root ganglia: 54% of beta3 small/medium neurons were NGF receptor trkA negative. Unlike beta1- and beta2, beta3-immunoreactivity did not decrease after avulsion injury, and the beta3:neurofilament ratio was significantly increased in proximal injured human nerves. beta3-subunit expression may thus be regulated differently from beta1, beta2 and Nav1.8. Targeting beta3 interactions with key alpha-subunits, particularly Nav1.3 and Nav1.8, may provide novel selective analgesics.

Publication types

  • Comparative Study

MeSH terms

  • Adult
  • Aged
  • Blotting, Western / methods
  • Cell Line
  • Embryo, Mammalian
  • Ganglia, Spinal / cytology*
  • Ganglia, Spinal / injuries
  • Gene Expression Regulation*
  • Humans
  • Immunohistochemistry / methods
  • Neurofilament Proteins / metabolism
  • Neurons, Afferent / metabolism*
  • Protein Subunits / genetics
  • Protein Subunits / metabolism*
  • Sodium Channels / genetics
  • Sodium Channels / metabolism*
  • Time Factors
  • Transfection / methods

Substances

  • Neurofilament Proteins
  • Protein Subunits
  • Sodium Channels