Tyrosine kinase 2 interacts with and phosphorylates receptor for activated C kinase-1, a WD motif-containing protein

J Immunol. 2004 Jul 15;173(2):1151-7. doi: 10.4049/jimmunol.173.2.1151.

Abstract

Receptor for activated C kinase (Rack)-1 is a protein kinase C-interacting protein, and contains a WD repeat but has no enzymatic activity. In addition to protein kinase C, Rack-1 also binds to Src, phospholipase Cgamma, and ras-GTPase-activating proteins. Thus, Rack-1 is thought to function as a scaffold protein that recruits specific signaling elements. In a cytokine signaling cascade, Rack-1 has been reported to interact with the IFN-alphabeta receptor and Stat1. In addition, we show here that Rack-1 associates with a member of Jak, tyrosine kinase 2 (Tyk2). Rack-1 interacts weakly with the kinase domain and interacts strongly with the pseudokinase domain of Tyk2. Rack-1 associates with Tyk2 via two regions, one in the N terminus and one in the middle portion (aa 138-203) of Rack-1. Jak activation causes the phosphorylation of tyrosine 194 on Rack-1. After phosphorylation, Rack-1 is translocated toward the perinuclear region. In addition to functioning as a scaffolding protein, these results raise the possibility that Rack-1 functions as a signaling molecule in cytokine signaling cascades.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Motifs
  • Humans
  • Phosphorylation
  • Protein Structure, Tertiary
  • Protein-Tyrosine Kinases / metabolism*
  • Receptors for Activated C Kinase
  • Receptors, Cell Surface / metabolism*
  • TYK2 Kinase
  • Tyrosine / metabolism

Substances

  • Receptors for Activated C Kinase
  • Receptors, Cell Surface
  • Tyrosine
  • Protein-Tyrosine Kinases
  • TYK2 Kinase
  • TYK2 protein, human