Analgesic activity of anticancer agent suramin

Anticancer Drugs. 1992 Apr;3(2):91-4. doi: 10.1097/00001813-199204000-00003.

Abstract

Suramin exhibited morphine-like analgesic activity in mice. It antagonized both thermal (hot-plate) and acetic acid-evoked writhing responses with ED50 values 1/100 and 1/68, respectively, that of morphine. The suramin- and morphine-induced hot-plate analgesia was suppressed by administration of 0.5 mg/kg naloxone. However, lower doses (5-30 micrograms/kg) of naloxone produced dose-related potentiation or suppression of suramin and morphine analgesia. This potentiation effect may be due to the inhibition of writhing by naloxone itself rather than be a direct antagonism of the morphine effect.

MeSH terms

  • Analgesia
  • Analgesics / pharmacology*
  • Animals
  • Dose-Response Relationship, Drug
  • Male
  • Mice
  • Mice, Inbred ICR
  • Morphine
  • Naloxone
  • Pain Measurement
  • Suramin / pharmacology*

Substances

  • Analgesics
  • Naloxone
  • Suramin
  • Morphine