Effective antiplatelet therapy does not prolong transgenic pig to baboon cardiac xenograft survival

Xenotransplantation. 2004 Sep;11(5):436-43. doi: 10.1111/j.1399-3089.2004.00159.x.

Abstract

Background: Microvascular thrombosis is a prominent characteristic of delayed xenograft rejection, therefore the effects of antiplatelet therapy with aspirin and clopidogrel on long-term cardiac xenograft function was investigated in a heterotopic pig-to-baboon cardiac transplant model.

Methods: Donor hearts from human CD46 transgenic pigs were transplanted heterotopically to baboons. The recipients received immunosuppression that included tacrolimus, sirolimus, corticosteroids, anti-CD20 monoclonal antibody and TPC, an alpha-galactosyl-polyethylene glycol conjugate. In group 1 (n = 9) in addition to immunosuppression, the recipients received combination therapy consisting of aspirin (80 mg/day) and clopidogrel (75 mg/day) beginning 2 days after transplant and continuing until cessation of graft function. Antiaggregatory efficacy was evaluated by platelet aggregation assay. In group 2 (n = 9) antiplatelet drugs were not given.

Results: Functional assays confirmed inhibition of platelet aggregation in group 1 suggesting sufficient systemic effects of the treatment. However, anticoagulant therapy did not result in significant prolongation of xenograft function (group 1: median survival 22 days, range 15 to 30 days; group 2: median survival 15 days, range 4 to 53 days). Histologic analysis at rejection revealed no difference in the level of platelet containing thrombi between the groups.

Conclusions: Inhibition of platelet aggregation by a combination of aspirin and clopidogrel did not have a significant impact on the length of xenograft survival or on the development of microvascular thrombosis in this pig-to-primate model.

MeSH terms

  • Animals
  • Animals, Genetically Modified
  • Antigens, CD / genetics
  • Aspirin / pharmacology
  • Clopidogrel
  • Graft Rejection / immunology
  • Graft Rejection / pathology
  • Graft Survival / drug effects
  • Graft Survival / immunology*
  • Heart Transplantation / immunology*
  • Heart Transplantation / pathology
  • Humans
  • Membrane Cofactor Protein
  • Membrane Glycoproteins / genetics
  • Papio anubis
  • Platelet Aggregation / drug effects
  • Platelet Aggregation / physiology*
  • Platelet Aggregation Inhibitors / pharmacology*
  • Swine
  • Ticlopidine / analogs & derivatives*
  • Ticlopidine / pharmacology
  • Time Factors
  • Transplantation, Heterologous / immunology*
  • Transplantation, Heterologous / pathology

Substances

  • Antigens, CD
  • CD46 protein, human
  • Membrane Cofactor Protein
  • Membrane Glycoproteins
  • Platelet Aggregation Inhibitors
  • Clopidogrel
  • Ticlopidine
  • Aspirin