[Anticholinergic Effect of a New Antiarrhythmic Class III Drug RG-2]

Kardiologiia. 2004;44(7):62-6.
[Article in Russian]

Abstract

In experiments on isolated rat and rabbit right atrium, a new class III antiarrhythmic drug RG-2 (0,01-1 microM) was shown to have anticholinergic action competing with 0.2-1 mM carbachol. RG-2 (0.1-1 microM) produced dose-dependent increase of APD90% in rat and rabbit atrial cells and had no effects on other action potential parameters. In presence of carbachol RG-2 produced significantly greater increase of APD90% and caused significant increase of APD50%. Thus RG-2 exerts anticholinergic action, which can take important part in RG-2 antiarrhythmic activity.

MeSH terms

  • Action Potentials / drug effects
  • Animals
  • Anti-Arrhythmia Agents* / pharmacology
  • Cholinergic Antagonists
  • Heart Atria* / drug effects

Substances

  • Anti-Arrhythmia Agents
  • Cholinergic Antagonists