[Killing effect of adenovirus mediated fusion gene cytosine and deaminase uracil phosphoribosyl transferase directed by glutathione S-transferase P1 promoter on cisplatin-resistant ovarian cancer cells in vitro]

Zhonghua Fu Chan Ke Za Zhi. 2004 Jul;39(7):478-81.
[Article in Chinese]

Abstract

Objective: To construct an adenoviral vector in which the fusion gene cytosine and uracil phosphoribosyl (UPP) transferase was directed by glutathione S-transferase P1 (GSTP1) promoter, and to investigate specific killing effect of the suicide gene system on cisplatin-resistant ovarian cancer cells.

Methods: Recombinant adenovirus was generated through homologous recombination in bacteria. A2780 and A2780/DDP cells were infected with Ad and then received flucytosine (5-FC) administration. The relative survival of these cells was tested. And a bystander effect was observed by mixing gene-transferred and gene-untransferred A2780/DDP cells with 5-FC.

Results: In vitro, when MOI was 100 and 5-FC was 250 micro g/ml, relative survival rate of A2780/DDP cells was only (3.6 +/- 1.0)%; that of A2780 cells was (76.5 +/- 2.8)%. Significant bystander effect was caused by CD-UPP gene and 20% gene-transferred A2780/DDP cells induced 80.3% of total cells to death.

Conclusion: Recombinant adenovirus carrying CD-UPP gene driven by GSTP1 promoter has a specific killing effect on cisplatin-resistant ovarian cancer cells.

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenoviruses, Human / genetics
  • Antineoplastic Agents / pharmacology
  • Cisplatin / pharmacology*
  • Cytosine Deaminase / genetics*
  • Drug Resistance, Neoplasm
  • Female
  • Flucytosine / therapeutic use
  • Genetic Therapy
  • Glutathione S-Transferase pi
  • Glutathione Transferase / genetics*
  • Humans
  • Isoenzymes / genetics*
  • Ovarian Neoplasms / pathology*
  • Pentosyltransferases / genetics*
  • Pentosyltransferases / metabolism
  • Promoter Regions, Genetic
  • Recombinant Fusion Proteins / genetics
  • Recombinant Fusion Proteins / metabolism
  • Transfection
  • Tumor Cells, Cultured

Substances

  • Antineoplastic Agents
  • Isoenzymes
  • Recombinant Fusion Proteins
  • Flucytosine
  • Pentosyltransferases
  • uracil phosphoribosyltransferase
  • GSTP1 protein, human
  • Glutathione S-Transferase pi
  • Glutathione Transferase
  • Cytosine Deaminase
  • Cisplatin