Disruption of cell-cell contact maximally but transiently activates AhR-mediated transcription in 10T1/2 fibroblasts

Toxicol Appl Pharmacol. 2004 Sep 15;199(3):220-38. doi: 10.1016/j.taap.2003.12.025.

Abstract

The aryl hydrocarbon receptor (AhR) is activated by 2,3,7,8-tetrachlorodibenzo-p-dioxin (TCDD), but activation without an exogenous ligand also occurs when normal cell-cell contact is prevented. Suspension of several C3H10T1/2 fibroblast clonal sub-lines that contain an integrated AhR-responsive reporter produced a time course and level of reporter activation and CYP1B1 induction that paralleled TCDD stimulation in confluent monolayer culture. Suspension activation was, however, more transient. Loss of cell-cell contact at low density also activated these reporters independent of cell cycle changes to levels comparable to TCDD stimulation of confluent cells. Loss of cell-cell contact may, therefore, activate AhR. Suspension and TCDD activations exhibited comparable nuclear translocation of AhR and then AhR/ARNT complex formation. Each AhR activation process was equally attenuated by inhibition of, respectively, HSP90 ATPase, the 26S proteosome, and by depletion of intracellular Ca2+. By contrast, the AhR antagonist alpha-naphthoflavone (alphaNF) blocked ligand-stimulated AhR activity, but not activation through loss of cell-cell contact. Suspension-induced reporter activation was selectively enhanced by LiCl, which prevented GSK-3beta effects on the simultaneously released beta-catenin. The effects of suspension and LiCl on reporters were reversed by Ro-31-8220, which did not affect beta-catenin, TCDD-activation processes, or AhR turnover. Neither LiCl nor Ro-31-8220 altered suspension-induced AhR/ARNT complex formation. Loss of cell-cell contact permits nuclear translocation and AhR activation that is largely replicated after TCDD binding, but with activity differences due to contact-sensitive factors functioning after AhR/ARNT complex formation.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Aryl Hydrocarbon Hydroxylases / biosynthesis
  • Aryl Hydrocarbon Hydroxylases / genetics
  • Cell Adhesion / drug effects
  • Cell Communication / physiology*
  • Cell Differentiation / drug effects
  • Cell Division / physiology
  • Cell Line
  • Cell Nucleus / drug effects
  • Cell Nucleus / ultrastructure
  • Culture Media
  • Cytochrome P-450 CYP1B1
  • Cytoskeletal Proteins / metabolism
  • Electrophoretic Mobility Shift Assay
  • Environmental Pollutants / pharmacology
  • Fibroblasts / metabolism*
  • Fibroblasts / physiology*
  • Gene Expression Regulation, Enzymologic / genetics
  • Genes, Reporter
  • Immunoblotting
  • Lithium Chloride / pharmacology
  • Luciferases / genetics
  • Methylcellulose
  • Mice
  • Mice, Inbred C3H
  • Polychlorinated Dibenzodioxins / pharmacology
  • Protein Transport
  • Receptors, Aryl Hydrocarbon / antagonists & inhibitors
  • Receptors, Aryl Hydrocarbon / biosynthesis*
  • Receptors, Aryl Hydrocarbon / genetics*
  • Trans-Activators / metabolism
  • Transcription, Genetic / physiology*
  • beta Catenin

Substances

  • CTNNB1 protein, mouse
  • Culture Media
  • Cytoskeletal Proteins
  • Environmental Pollutants
  • Polychlorinated Dibenzodioxins
  • Receptors, Aryl Hydrocarbon
  • Trans-Activators
  • beta Catenin
  • Methylcellulose
  • Luciferases
  • Aryl Hydrocarbon Hydroxylases
  • Cyp1b1 protein, mouse
  • Cytochrome P-450 CYP1B1
  • Lithium Chloride