Up-regulated neuronal nitric oxide synthase compensates coronary flow response to bradykinin in endothelial nitric oxide synthase-deficient mice

J Cardiovasc Pharmacol. 2004 Oct;44(4):437-45. doi: 10.1097/01.fjc.0000139450.64337.cd.

Abstract

It has been reported that endothelium-dependent relaxations are preserved in isolated coronary arteries of endothelial nitric oxide synthase-deficient (eNOS-/-) mice with a possible involvement of nNOS. However, it remains to be examined whether nNOS compensates coronary flow response in a beating heart of eNOS-/- mice and if so, whether and where nNOS is up-regulated. Coronary flow response to bradykinin was examined in Langendorff-perfused hearts from WT and eNOS-/- mice. Bradykinin-induced coronary flow was greater in eNOS-/- mice than in WT mice, and indomethacin had no inhibitory effect on it. Bradykinin receptor antagonist HOE-140 abolished the bradykinin response in both strains. Non-selective NOSs inhibitor L-NNA inhibited the bradykinin-induced coronary flow in both strains, whereas specific inhibitors of nNOS, SMTC, and 7-NI, significantly attenuated the coronary flow response only in eNOS-/- mice. A guanylate cyclase inhibitor ODQ also attenuated the bradykinin response in eNOS-/- mice. Immunohistochemistry revealed the presence of nNOS mainly in coronary vascular smooth muscle cells (VSMCs) in both strains and Western blot analysis demonstrated a marked increase in cardiac nNOS expression in eNOS-/- mice. These results indicate that nNOS compensates coronary flow response to bradykinin in eNOS-/- mice, for which up-regulation of nNOS in VSMCs may be involved.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Bradykinin / analogs & derivatives*
  • Bradykinin / pharmacology*
  • Bradykinin / physiology
  • Citrulline / analogs & derivatives*
  • Citrulline / pharmacology
  • Coronary Circulation / physiology
  • Coronary Vessels / drug effects
  • Coronary Vessels / enzymology
  • Enzyme Inhibitors / pharmacology
  • Female
  • Immunohistochemistry
  • In Vitro Techniques
  • Indomethacin / pharmacology
  • Male
  • Mice
  • Mice, Knockout
  • Nerve Tissue Proteins / antagonists & inhibitors
  • Nerve Tissue Proteins / biosynthesis
  • Neurons / enzymology
  • Neurons / metabolism*
  • Nitric Oxide Synthase / antagonists & inhibitors
  • Nitric Oxide Synthase / biosynthesis
  • Nitric Oxide Synthase / genetics*
  • Nitric Oxide Synthase Type I
  • Nitric Oxide Synthase Type II
  • Nitric Oxide Synthase Type III
  • Nitroarginine / pharmacology
  • Oxadiazoles / pharmacology
  • Thiourea / analogs & derivatives*
  • Thiourea / pharmacology
  • Up-Regulation*
  • Vasodilation / physiology

Substances

  • 1H-(1,2,4)oxadiazolo(4,3-a)-quiloxalin-1-one
  • Enzyme Inhibitors
  • Nerve Tissue Proteins
  • Oxadiazoles
  • Nitroarginine
  • Citrulline
  • icatibant
  • Nitric Oxide Synthase
  • Nitric Oxide Synthase Type I
  • Nitric Oxide Synthase Type II
  • Nitric Oxide Synthase Type III
  • Nos1 protein, mouse
  • Nos3 protein, mouse
  • Thiourea
  • S-methylthiocitrulline
  • Bradykinin
  • Indomethacin