Phytosphingosine in combination with ionizing radiation enhances apoptotic cell death in radiation-resistant cancer cells through ROS-dependent and -independent AIF release

Blood. 2005 Feb 15;105(4):1724-33. doi: 10.1182/blood-2004-07-2938. Epub 2004 Oct 14.

Abstract

The use of chemical modifiers as radiosensitizers in combination with low-dose irradiation may increase the therapeutic effect on cancer by overcoming a high apoptotic threshold. Here, we showed that phytosphingosine treatment in combination with gamma-radiation enhanced apoptotic cell death of radiation-resistant human T-cell lymphoma in a caspase-independent manner. Combination treatment induced an increase in intracellular reactive oxygen species (ROS) level, mitochondrial relocalization of B-cell lymphoma-2(Bcl-2)-associated X protein (Bax), poly-adenosine diphosphate (ADP)-ribose polymerase 1 (PARP-1) activation, and nuclear translocation of apoptosis-inducing factor (AIF). siRNA targeting of AIF effectively protected cells from the combination treatment-induced cell death. An antioxidant, N-acetyl-L-cysteine (NAC), inhibited Bax relocalization and AIF translocation but not PARP-1 activation. Moreover, transfection of Bax-siRNA significantly inhibited AIF translocation. Pretreatment of PARP-1 inhibitor, DPQ (3,4-dihydro-5-[4-(1-piperidinyl)-butoxy]-1(2H)-isoquinolinone), or PARP-1-siRNA also partially attenuated AIF translocation, whereas the same treatment did not affect intracellular ROS level and Bax redistribution. Taken together, these results demonstrate that enhancement of cell death of radiation-resistant cancer cells by phytosphingosine treatment in combination with gamma-radiation is mediated by nuclear translocation of AIF, which is in turn mediated both by ROS-dependent Bax relocalization and ROS-independent PARP-1 activation. The molecular signaling pathways that we elucidated in this study may provide potential drug targets for radiation sensitization of cancers refractive to radiation therapy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Active Transport, Cell Nucleus / drug effects
  • Active Transport, Cell Nucleus / radiation effects
  • Apoptosis / drug effects*
  • Apoptosis / radiation effects*
  • Apoptosis Inducing Factor
  • Cell Nucleus / drug effects
  • Cell Nucleus / metabolism
  • Cell Nucleus / radiation effects
  • Clone Cells
  • Combined Modality Therapy
  • Enzyme Activation / drug effects
  • Enzyme Activation / radiation effects
  • Flavoproteins / metabolism*
  • Gamma Rays*
  • Humans
  • Intracellular Membranes / drug effects
  • Intracellular Membranes / metabolism
  • Intracellular Membranes / radiation effects
  • Jurkat Cells
  • Membrane Potentials / drug effects
  • Membrane Potentials / radiation effects
  • Membrane Proteins / metabolism*
  • Mitochondria / drug effects
  • Mitochondria / metabolism
  • Mitochondria / radiation effects
  • Poly(ADP-ribose) Polymerases / metabolism
  • Proto-Oncogene Proteins c-bcl-2 / metabolism
  • Radiation Tolerance*
  • Reactive Oxygen Species / pharmacology*
  • Sphingosine / analogs & derivatives*
  • Sphingosine / pharmacology*
  • bcl-2-Associated X Protein

Substances

  • AIFM1 protein, human
  • Apoptosis Inducing Factor
  • BAX protein, human
  • Flavoproteins
  • Membrane Proteins
  • Proto-Oncogene Proteins c-bcl-2
  • Reactive Oxygen Species
  • bcl-2-Associated X Protein
  • Poly(ADP-ribose) Polymerases
  • phytosphingosine
  • Sphingosine