Oxiracetam antagonizes the disruptive effects of scopolamine on memory in the radial maze

Psychopharmacology (Berl). 1992;106(2):175-8. doi: 10.1007/BF02801969.

Abstract

The effects exerted by oxiracetam on the disruption of performance induced by scopolamine in the radial arm maze were investigated in overtrained rats. Scopolamine induced a dose-related decrease in the efficiency of responding and an increase of running time. The effect of the SC injection of 0.2 mg/kg scopolamine on the efficiency of responding was antagonized by the IP administration of 30 mg/kg oxiracetam, while the effect on running time induced by the same dose of scopolamine was not. Physostigmine (0.3 mg/kg SC) antagonized both effects of 0.2 mg/kg scopolamine. Methylscopolamine, at the dose of 0.2 mg/kg SC, was devoid of any effect on both parameters. Increasing the dose of methylscopolamine to 0.63 mg/kg did cause serious peripheral effects which eventually prevented some animals from completing the task. Similar peripheral effects were observed after administration of 0.63 mg/kg scopolamine. The effects of this dose of scopolamine on efficiency and running time were not antagonized by pretreatment with 100 mg/kg oxiracetam. Oxiracetam alone (30 or 100 mg/kg IP) did not modify the performance of previously trained rats. The present results suggest that oxiracetam selectively restores cholinergic mechanisms which are involved in learning and memory.

MeSH terms

  • Animals
  • Dose-Response Relationship, Drug
  • Male
  • Memory / drug effects*
  • Motor Activity / drug effects
  • N-Methylscopolamine
  • Parasympathetic Nervous System / drug effects
  • Parasympatholytics / pharmacology
  • Physostigmine / pharmacology
  • Psychotropic Drugs / pharmacology*
  • Pyrrolidines / pharmacology*
  • Rats
  • Rats, Inbred Strains
  • Scopolamine / antagonists & inhibitors*
  • Scopolamine / pharmacology
  • Scopolamine Derivatives / pharmacology

Substances

  • Parasympatholytics
  • Psychotropic Drugs
  • Pyrrolidines
  • Scopolamine Derivatives
  • Physostigmine
  • Scopolamine
  • oxiracetam
  • N-Methylscopolamine