c-kit Expression in small cell carcinoma of the urinary bladder: prognostic and therapeutic implications

Mod Pathol. 2005 Mar;18(3):320-3. doi: 10.1038/modpathol.3800318.

Abstract

The prognosis for small cell carcinoma of the urinary bladder is poor, and strategies for improved therapy are needed. Targeted therapy against the c-kit proto-oncogene has been successful in the management of gastrointestinal stromal tumor. We investigated the expression of c-kit in 52 cases of small cell carcinoma of the urinary bladder. Specimens with more than 10% of cells demonstrating strong membrane staining were considered to have positive immunostaining for c-kit. c-kit expression was detected in 21 of 52 specimens from these patients. Among the 21 specimens, seven had less than 10% staining, and were considered to be negative. Nine had 11-50% staining, and five had more than 50% staining. Overall, 14 of 52 (27%) small cell carcinomas of the urinary bladder were positive for c-kit expression. During a median follow-up of 11 months, 60% of the patients died of bladder cancer. No association was found between c-kit expression and survival or other clinicopathologic parameters. Five-year cancer-specific survivals for c-kit-positive and c-kit-negative tumors were 9 and 15%, respectively (P=0.36). A significant proportion (27%) of small cell carcinomas of the urinary bladder expressed c-kit, suggesting that it may prove useful as a therapeutic target in small cell carcinoma of the urinary bladder.

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Benzamides
  • Carcinoma, Small Cell / metabolism
  • Carcinoma, Small Cell / pathology*
  • Female
  • Follow-Up Studies
  • Humans
  • Imatinib Mesylate
  • Immunohistochemistry
  • Male
  • Middle Aged
  • Piperazines / therapeutic use
  • Prognosis
  • Protein Kinase Inhibitors / therapeutic use
  • Proto-Oncogene Mas
  • Proto-Oncogene Proteins c-kit / biosynthesis*
  • Pyrimidines / therapeutic use
  • Survival Analysis
  • Urinary Bladder / drug effects
  • Urinary Bladder / metabolism
  • Urinary Bladder / pathology
  • Urinary Bladder Neoplasms / metabolism
  • Urinary Bladder Neoplasms / pathology*

Substances

  • Benzamides
  • MAS1 protein, human
  • Piperazines
  • Protein Kinase Inhibitors
  • Proto-Oncogene Mas
  • Pyrimidines
  • Imatinib Mesylate
  • Proto-Oncogene Proteins c-kit