Early growth response-1 regulates lipopolysaccharide-induced suppressor of cytokine signaling-1 transcription

J Biol Chem. 2005 Jan 28;280(4):2596-605. doi: 10.1074/jbc.M408938200. Epub 2004 Nov 15.

Abstract

Suppressor of cytokine signaling (SOCS)-1 is a critical regulator of lipopolysaccharide (LPS) tolerance and LPS-induced cytokine production. The mechanisms regulating the transcription of SOCS-1 in response to LPS are not entirely understood. Functional analysis of the SOCS-1 promoter demonstrates that early growth response-1 (Egr-1) is an important transcriptional regulator of SOCS-1. Two Egr-1 binding sites are present within the SOCS-1 promoter as shown by EMSA and supershift analysis. Further, mutation of the Egr-1 binding sites significantly reduces both the basal and LPS-induced transcriptional activity of the promoter. Chromatin immunoprecipitation experiments confirm LPS-induced binding of Egr-1 to the SOCS-1 promoter in vivo. Additionally, Egr-1(-/-) macrophages show reduced levels of LPS-induced SOCS-1 expression in comparison with macrophages derived from Egr-1(+/+) littermate controls. These results demonstrate an important role for Egr-1 in regulating both the basal and LPS-induced activity of the SOCS-1 promoter.

MeSH terms

  • Animals
  • Base Sequence
  • Binding Sites
  • Blotting, Northern
  • Cell Line
  • Chromatin Immunoprecipitation
  • Codon
  • DNA-Binding Proteins / physiology*
  • Early Growth Response Protein 1
  • Gene Expression Regulation
  • Humans
  • Immediate-Early Proteins / physiology*
  • Intracellular Signaling Peptides and Proteins / chemistry
  • Lipopolysaccharides / metabolism*
  • Luciferases / metabolism
  • Macrophages / metabolism
  • Mice
  • Mice, Transgenic
  • Molecular Sequence Data
  • Mutation
  • Plasmids / metabolism
  • Promoter Regions, Genetic
  • Protein Binding
  • RNA, Messenger / metabolism
  • Repressor Proteins / biosynthesis*
  • Repressor Proteins / chemistry
  • Sequence Homology, Nucleic Acid
  • Suppressor of Cytokine Signaling 1 Protein
  • Suppressor of Cytokine Signaling Proteins
  • Transcription Factors / physiology*
  • Transcription, Genetic
  • Transgenes

Substances

  • Codon
  • DNA-Binding Proteins
  • EGR1 protein, human
  • Early Growth Response Protein 1
  • Immediate-Early Proteins
  • Intracellular Signaling Peptides and Proteins
  • Lipopolysaccharides
  • RNA, Messenger
  • Repressor Proteins
  • SOCS1 protein, human
  • Suppressor of Cytokine Signaling 1 Protein
  • Suppressor of Cytokine Signaling Proteins
  • Transcription Factors
  • Luciferases