Analysis of SHP-1-mediated down-regulation of the TRK-T3 oncoprotein identifies Trk-fused gene (TFG) as a novel SHP-1-interacting protein

J Biol Chem. 2005 Feb 4;280(5):3382-9. doi: 10.1074/jbc.M407522200. Epub 2004 Nov 22.

Abstract

SHP-1 is a cytoplasmic SH2 domain containing protein-tyrosine phosphatase (PTP) involved in the negative regulation of multiple signaling pathways in hematopoietic, nervous, and epithelial cells. The thyroid TRK-T3 oncogene consists of the NTRK1 tyrosine kinase domain fused in-frame with sequences of the TFG (TRK-fused gene), encoding a protein of unknown function. TFG contains a coiled-coil domain responsible for TRK-T3 oligomerization. In addition, recent analysis of the sequences outside of the coiled-coil domain suggested possible interactions with other proteins. Based on the presence of a putative SHP-1 SH2-binding site within the TFG sequences, we have investigated the role of the SHP-1 phosphatase in TRK-T3 oncoprotein signaling. In this study we show that SHP-1 interacts with and down-regulates TRK-T3. We provide evidence that SHP-1 SH2 and catalytic domains, respectively, associate with the TFG- and NTRK1-derived portions of TRK-T3. Our data contribute to the definition of cellular mechanisms involved in thyroid tumorigenesis. Moreover, it reveals TFG as a novel protein able to modulate SHP-1 activity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Catalysis
  • Down-Regulation / physiology
  • Enzyme Activation / physiology
  • Humans
  • Intracellular Signaling Peptides and Proteins
  • Kidney / cytology
  • Mice
  • Mutagenesis
  • NIH 3T3 Cells
  • Protein Structure, Tertiary
  • Protein Tyrosine Phosphatase, Non-Receptor Type 6
  • Protein Tyrosine Phosphatases / chemistry
  • Protein Tyrosine Phosphatases / genetics*
  • Protein Tyrosine Phosphatases / metabolism*
  • Proteins / chemistry
  • Proteins / genetics*
  • Proteins / metabolism*
  • Receptor, trkA / chemistry
  • Receptor, trkA / genetics
  • Receptor, trkA / metabolism
  • Thyroid Neoplasms / physiopathology
  • Tyrosine / metabolism

Substances

  • Intracellular Signaling Peptides and Proteins
  • Proteins
  • TFG protein, human
  • Tyrosine
  • Receptor, trkA
  • PTPN6 protein, human
  • Protein Tyrosine Phosphatase, Non-Receptor Type 6
  • Protein Tyrosine Phosphatases
  • Ptpn6 protein, mouse