The effects of intracellular Ca2+ on cardiac K+ channel expression and activity: novel insights from genetically altered mice

J Physiol. 2005 Feb 1;562(Pt 3):745-58. doi: 10.1113/jphysiol.2004.076216. Epub 2004 Nov 25.

Abstract

We tested the hypothesis that chronic changes in intracellular Ca(2+) (Ca(2+)(i)) can result in changes in ion channel expression; this represents a novel mechanism of crosstalk between changes in Ca(2+) cycling proteins and the cardiac action potential (AP) profile. We used a transgenic mouse with cardiac-specific overexpression of sarcoplasmic reticulum Ca(2+) ATPase (SERCA) isoform 1a (SERCA1a OE) with a significant alteration of SERCA protein levels without cardiac hypertrophy or failure. Here, we report significant changes in the expression of a transient outward K(+) current (I(to,f)), a slowly inactivating K(+) current (I(K,slow)) and the steady state current (I(SS)) in the transgenic mice with resultant prolongation in cardiac action potential duration (APD) compared with the wild-type littermates. In addition, there was a significant prolongation of the QT interval on surface electrocardiograms in SERCA1a OE mice. The electrophysiological changes, which correlated with changes in Ca(2+)(i), were further corroborated by measuring the levels of ion channel protein expression. To recapitulate the in vivo experiments, the effects of changes in Ca(2+)(i) on ion channel expression were further tested in cultured adult and neonatal mouse cardiac myocytes. We conclude that a primary defect in Ca(2+) handling proteins without cardiac hypertrophy or failure may produce profound changes in K(+) channel expression and activity as well as cardiac AP.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Action Potentials / physiology*
  • Animals
  • Calcium / metabolism*
  • Calcium-Transporting ATPases / genetics
  • Calcium-Transporting ATPases / metabolism*
  • Cells, Cultured
  • Electrocardiography
  • Enzyme Activation
  • Gene Expression Regulation, Enzymologic / physiology*
  • Heart Ventricles / cytology
  • Heart Ventricles / embryology
  • Heart Ventricles / metabolism
  • Intracellular Fluid / metabolism
  • Ion Channel Gating / physiology*
  • Mice
  • Mice, Transgenic / metabolism*
  • Muscle Cells / physiology*
  • Recombinant Proteins / metabolism
  • Sarcoplasmic Reticulum Calcium-Transporting ATPases

Substances

  • Recombinant Proteins
  • Sarcoplasmic Reticulum Calcium-Transporting ATPases
  • Calcium-Transporting ATPases
  • Calcium