Aminothiazole inhibitors of HCV RNA polymerase

Bioorg Med Chem Lett. 2005 Jan 3;15(1):115-9. doi: 10.1016/j.bmcl.2004.10.024.

Abstract

Aminothiazole-based inhibitors designed for HCV polymerase display low micromolar potencies in biochemical assays. These compounds show a stringent preference for a cyclohexyl hydrophobe at the 2-amino position. The composition of these compounds suggests that they may be interacting at a recently discovered allosteric site on the polymerase.

MeSH terms

  • DNA-Directed RNA Polymerases / antagonists & inhibitors*
  • Enzyme Inhibitors / chemical synthesis
  • Enzyme Inhibitors / pharmacology*
  • Hepacivirus / enzymology*
  • Thiazoles / chemical synthesis
  • Thiazoles / pharmacology*

Substances

  • Enzyme Inhibitors
  • Thiazoles
  • DNA-Directed RNA Polymerases