Cyclooxygenase-2 selective inhibitor prevents implantation of eutopic endometrium to ectopic sites in rats

Fertil Steril. 2004 Dec;82(6):1609-15. doi: 10.1016/j.fertnstert.2004.07.946.

Abstract

Objective: To evaluate Cox-2 inhibition on surgically induced endometriosis in rats.

Design: Prospective, randomized study

Setting: Academic facility.

Animal(s): Seventy adult female Sprague-Dawley rats.

Intervention(s): Uterine fragments were implanted into abdominal peritoneum with suture (site A), and/or into the pelvic cavity without suture (site B). Oral gavage of Cox-2 inhibitor (5 mg/kg/day, twice/day) was started 4 weeks postimplantation (protocol-1), after implantation (protocol-2), or beforehand (protocol-3). Controls received vehicle. Immunohistochemistry evaluated Cox-2 expression after treatment.

Main outcome measurement(s): Presence and size of ectopic implants after treatment.

Result(s): Protocol-1: After 4 weeks' treatment, size of ectopic implants (site A) was significantly reduced compared with pretreatment size. After 8 weeks' treatment, no ectopic implants were detected in 2 (40%, site A) and 3 (60%, site B) rats. Protocol-2: After 2 weeks' treatment, no ectopic implants were detected in 3 (50%, site A) and 2 (33%, site B) rats. After 4 weeks' treatment, no ectopic implants were detected in 3 (50%, site A) and 3 (50%, site B) rats. Protocol-3: After 2 or 4 weeks' vehicle-only treatment, ectopic implants were in all rats (site B).

Conclusion(s): Cox-2 selective inhibition was effective in a rat model of endometriosis, particularly in prevention of ectopic implants.

MeSH terms

  • Animals
  • Cyclooxygenase 2
  • Cyclooxygenase 2 Inhibitors
  • Cyclooxygenase Inhibitors / administration & dosage
  • Cyclooxygenase Inhibitors / pharmacology*
  • Disease Models, Animal
  • Drug Administration Schedule
  • Endometriosis / enzymology
  • Endometriosis / pathology
  • Endometriosis / prevention & control*
  • Female
  • Immunohistochemistry
  • Isoenzymes / antagonists & inhibitors*
  • Isoenzymes / metabolism
  • Prostaglandin-Endoperoxide Synthases / metabolism
  • Random Allocation
  • Rats
  • Rats, Sprague-Dawley

Substances

  • Cyclooxygenase 2 Inhibitors
  • Cyclooxygenase Inhibitors
  • Isoenzymes
  • Cyclooxygenase 2
  • Prostaglandin-Endoperoxide Synthases