T cell receptor-induced activation of phospholipase C-gamma1 depends on a sequence-independent function of the P-I region of SLP-76

J Biol Chem. 2005 Mar 4;280(9):8364-70. doi: 10.1074/jbc.M409437200. Epub 2004 Dec 28.

Abstract

SLP-76 forms part of a hematopoietic-specific adaptor protein complex, and is absolutely required for T cell development and activation. T cell receptor (TCR)-induced activation of phospholipase C-gamma1 (PLC-gamma1) depends on three features of SLP-76: the N-terminal tyrosine phosphorylation sites, the Gads-binding site, and an intervening sequence, denoted the P-I region, which binds to the SH3 domain of PLC-gamma1 (SH3(PLC)) via a low affinity interaction. Despite extensive research, the mechanism whereby SLP-76 regulates PLC-gamma1 remains uncertain. In this study, we uncover and explore an apparent paradox: whereas the P-I region as a whole is essential for TCR-induced activation of PLC-gamma1 and nuclear factor of activated T cells (NFAT), no particular part of this region is absolutely required. To better understand the contribution of the P-I region to PLC-gamma1 activation, we mapped the PLC-gamma1-binding site within the region, and created a SLP-76 mutant that fails to bind SH3(PLC), but is fully functional, mediating TCR-induced phosphorylation of PLC-gamma1 at tyrosine 783, calcium flux, and nuclear factor of activated T cells activation. Unexpectedly, full functionality of this mutant was maintained even under less than optimal stimulation conditions, such as a low concentration of the anti-TCR antibody. Another SLP-76 mutant, in which the P-I region was scrambled to abolish any sequence-dependent protein-binding motifs, also retained significant functionality. Our results demonstrate that SLP-76 need not interact with SH3(PLC) to activate PLC-gamma1, and further suggest that the P-I region of SLP-76 serves a structural role that is sequence-independent and is not directly related to protein-protein interactions.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adaptor Proteins, Signal Transducing
  • Alleles
  • Amino Acid Motifs
  • Binding Sites
  • Calcium / metabolism
  • Cell Line
  • Epitopes / chemistry
  • Gene Deletion
  • Genes, Reporter
  • Glutathione Transferase / metabolism
  • Humans
  • Immunoprecipitation
  • Jurkat Cells
  • Luciferases / metabolism
  • Mutation
  • Phospholipase C gamma
  • Phosphoproteins / chemistry*
  • Phosphoproteins / physiology*
  • Proline / chemistry
  • Protein Structure, Tertiary
  • Receptors, Antigen, T-Cell / metabolism*
  • Recombinant Fusion Proteins / metabolism
  • Structure-Activity Relationship
  • Time Factors
  • Transfection
  • Type C Phospholipases / metabolism*
  • src Homology Domains

Substances

  • Adaptor Proteins, Signal Transducing
  • Epitopes
  • Phosphoproteins
  • Receptors, Antigen, T-Cell
  • Recombinant Fusion Proteins
  • SLP-76 signal Transducing adaptor proteins
  • Proline
  • Luciferases
  • Glutathione Transferase
  • Type C Phospholipases
  • Phospholipase C gamma
  • Calcium