Enantioselective alkylations of tributyltin enolates catalyzed by Cr(salen)Cl: access to enantiomerically enriched all-carbon quaternary centers

J Am Chem Soc. 2005 Jan 12;127(1):62-3. doi: 10.1021/ja043601p.

Abstract

The catalytic asymmetric alpha-alkylation of tributyltin enolates with a range of primary alkyl halides is catalyzed by a chiral Cr(salen) complex. The reaction constitutes the first transition-metal-catalyzed system for alpha-alkylation of carbonyl substrates with this important class of electrophiles, providing access to five-, six-, and seven-membered ring ketone products bearing alpha-quaternary stereocenters in high enantioselectivity and synthetically useful yields.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Alkenes / chemistry*
  • Alkylation
  • Catalysis
  • Chromium / chemistry*
  • Ethylenediamines / chemistry*
  • Ketones / chemical synthesis*
  • Organometallic Compounds / chemistry*
  • Stereoisomerism
  • Trialkyltin Compounds / chemistry*

Substances

  • Alkenes
  • Ethylenediamines
  • Ketones
  • Organometallic Compounds
  • Trialkyltin Compounds
  • Chromium
  • tributyltin
  • disalicylaldehyde ethylenediamine