Migration of vascular smooth muscle cells by phospholipase A2 via specific binding sites

Biochim Biophys Acta. 1992 Apr 23;1125(2):210-4. doi: 10.1016/0005-2760(92)90047-y.

Abstract

Pancreatic-type group I phospholipase A2 (PLA2-I), EC 3.1.1.4, long thought to act as a digestive enzyme, has a specific binding site in several types of tissues and cells and these sites promote PLA2-I-stimulated DNA synthesis. In this study we report a PLA2-I action on the migration of rat embryonic thoracic aorta smooth muscle cells (A7r5). A7r5 cells had a single class of PLA2-I binding site with an equilibrium binding constant (Kd) value of 1.7 nM and a maximum binding capacity (Bmax) of 40,000 sites/cell. The migration activity of PLA2-I for A7r5 cells was examined using modified Boyden chambers. PLA2-I stimulated the migration dose-dependently, and the ED50 value was about 1 nM, which was almost the same as the Kd value for PLA2-I binding. Checkerboard analysis showed that the response of A7r5 cells to PLA2-I was chemokinetic, but not chemotactic. These findings reveal a new aspect of PLA2-I in the modulation of vascular function.

MeSH terms

  • 12-Hydroxy-5,8,10,14-eicosatetraenoic Acid
  • Animals
  • Aorta, Thoracic / embryology
  • Binding Sites
  • Cell Line
  • Cell Movement / drug effects*
  • Chemotactic Factors / pharmacology
  • Hydroxyeicosatetraenoic Acids / pharmacology
  • Interleukin-1 / pharmacology
  • Iodine Radioisotopes
  • Muscle, Smooth, Vascular / cytology
  • Muscle, Smooth, Vascular / enzymology
  • Muscle, Smooth, Vascular / physiology*
  • Phospholipases A / metabolism
  • Phospholipases A / physiology*
  • Phospholipases A2
  • Rats

Substances

  • Chemotactic Factors
  • Hydroxyeicosatetraenoic Acids
  • Interleukin-1
  • Iodine Radioisotopes
  • 12-Hydroxy-5,8,10,14-eicosatetraenoic Acid
  • Phospholipases A
  • Phospholipases A2