The positive regulation of human thyrotropin (TSH) receptor messenger ribonucleic acid by recombinant human TSH is at the intranuclear level

Endocrinology. 1992 May;130(5):2858-64. doi: 10.1210/endo.130.5.1572298.

Abstract

We have assessed the regulatory influence of human recombinant TSH (rec-hTSH) on its homologous receptor (TSHR) using a well characterized human fetal thyroid monolayer cell culture technique. Under the culture conditions employed, fetal human thyroid cells showed basal expression of TSHR-specific mRNA transcripts, and the addition of rec-hTSH (1 U/L) induced up to an 8-fold increase in specific mRNA over a 48-h observation period. This induction was simulated by bromo-cAMP in a dose-dependent manner, indicating that the stimulatory effect of rec-hTSH was active at the postreceptor level. Furthermore, there was no detectable increase in the transcription rate of the TSHR gene after stimulation with rec-hTSH for 12-36 h, although a marked increase in thyroglobulin-specific mRNA was observed. Rec-hTSH also had no influence on the half-life of TSHR-specific mRNA, which remained at approximately 16 h in the presence or absence of rec-hTSH. These data indicate that rec-hTSH induced up-regulation in human thyroid cell TSHR-specific mRNA and that the mechanism of this regulation was likely to be secondary to a posttranscriptional nuclear event involving changes in the regulation of primary unspliced mRNA for the TSHR.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 8-Bromo Cyclic Adenosine Monophosphate / pharmacology
  • Abortion, Spontaneous
  • Analysis of Variance
  • Base Sequence
  • Cell Nucleus / drug effects
  • Cell Nucleus / physiology*
  • Cells, Cultured
  • Dactinomycin / pharmacology
  • Female
  • Fetus
  • Gene Expression Regulation / drug effects*
  • Glyceraldehyde-3-Phosphate Dehydrogenases / genetics
  • Humans
  • Kinetics
  • Molecular Sequence Data
  • Monosaccharide Transport Proteins / genetics
  • Oligodeoxyribonucleotides
  • Polymerase Chain Reaction
  • Pregnancy
  • RNA, Messenger / analysis
  • RNA, Messenger / genetics*
  • RNA, Messenger / metabolism
  • Receptors, Thyrotropin / genetics*
  • Recombinant Proteins / pharmacology
  • Thyroid Gland / drug effects
  • Thyroid Gland / physiology*
  • Thyrotropin / pharmacology*
  • Transcription, Genetic / drug effects*

Substances

  • Monosaccharide Transport Proteins
  • Oligodeoxyribonucleotides
  • RNA, Messenger
  • Receptors, Thyrotropin
  • Recombinant Proteins
  • Dactinomycin
  • 8-Bromo Cyclic Adenosine Monophosphate
  • Thyrotropin
  • Glyceraldehyde-3-Phosphate Dehydrogenases