Surface modification of biodegradable polyesters with fatty acid conjugates for improved drug targeting

Biomaterials. 2005 Oct;26(28):5727-36. doi: 10.1016/j.biomaterials.2005.02.025. Epub 2005 Apr 18.

Abstract

We describe a general method for incorporating target ligands into the surface of biocompatible polyester poly(lactic-co-glycolic acid) (PLGA) 50/50 materials using fatty acids. Avidin-fatty acid conjugates were prepared and efficiently incorporated into PLGA. Avidin was chosen as an adaptor protein to facilitate the attachment of a variety of biotinylated ligands. We show that fatty acid preferentially associates with the hydrophobic PLGA matrix, rather than the external aqueous environment, facilitating a prolonged presentation of avidin over several weeks. We successfully applied this approach in both microspheres encapsulating a model protein, bovine serum albumin, and PLGA scaffolds fabricated by a salt-leaching method. Because of its ease, generality and flexibility, this strategy promises widespread utility in modifying the surface of PLGA-based materials for applications in drug delivery and tissue engineering.

Publication types

  • Evaluation Study
  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Absorbable Implants*
  • Avidin / administration & dosage
  • Avidin / analysis
  • Avidin / chemistry*
  • Coated Materials, Biocompatible / analysis
  • Coated Materials, Biocompatible / chemistry*
  • Diffusion
  • Drug Delivery Systems / methods*
  • Fatty Acids / chemistry*
  • Lactic Acid / analysis
  • Lactic Acid / chemistry*
  • Materials Testing
  • Microspheres
  • Particle Size
  • Polyesters / chemistry
  • Polyglycolic Acid / analysis
  • Polyglycolic Acid / chemistry*
  • Polylactic Acid-Polyglycolic Acid Copolymer
  • Polymers / analysis
  • Polymers / chemistry*
  • Surface Properties

Substances

  • Coated Materials, Biocompatible
  • Fatty Acids
  • Polyesters
  • Polymers
  • Avidin
  • Polylactic Acid-Polyglycolic Acid Copolymer
  • Polyglycolic Acid
  • Lactic Acid